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Synthesis of 1,2,3-Triazolyl Nucleoside Analogs as Potential Anti-Influenza A (H3N2 Subtype) Virus Agents.
Journal article   Peer reviewed

Synthesis of 1,2,3-Triazolyl Nucleoside Analogs as Potential Anti-Influenza A (H3N2 Subtype) Virus Agents.

Hanane Elayadi, Michael Smietana, Jean-Jacques Vasseur, Jan Balzarini and Hassan B. Lazrek
Archiv der Pharmazie / Chemistry in Life Sciences, Vol.347(2), pp.134-141
03/02/2014

Abstract

Anti-influenza A (H3N2) Click reaction 3-Triazolyl nucleoside
Montmorillonite K10 impregnated with copper dichloride and potassium iodide (CuCl2/KI/K10) was used as catalyst in the cycloaddition of azides and propargylnucleobases, to provide the corresponding 1,4-disubstituted 1,2,3-triazoles in good yield. All compounds 16-23 were evaluated for their antiviral activity in vitro. Compound 18 showed moderate inhibition against influenza virus A (H3N2).
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