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Synthesis and biological evaluation of 2-(3'-(1H-tetrazol-5-yl) bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mglu1 receptor antagonist
Article de revue   Avec comité de lecture

Synthesis and biological evaluation of 2-(3'-(1H-tetrazol-5-yl) bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mglu1 receptor antagonist

Gabriele Costantino, Katiuscia Maltoni, Maura Marinozzi, Emidio Camaioni, Laurent Prezeau, Jean-Philippe Pin et Roberto Pellicciari
Bioorganic & medicinal chemistry, Vol.9(2), pp.221-227
01/02/2001
PMID: 11249114

Résumé

Biological and medical sciences Glutamatergic system (aspartate and other excitatory aminoacids) Medical sciences Neuropharmacology Neurotransmitters. Neurotransmission. Receptors Pharmacology. Drug treatments

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