Logo image
Sign in
Synergistic Copper/Enamine Catalysis for the Regio-,Stereo-and Enantioselective Intermolecular α-Addition of Aldehydes to Allenamides
Journal article   Open access   Peer reviewed

Synergistic Copper/Enamine Catalysis for the Regio-,Stereo-and Enantioselective Intermolecular α-Addition of Aldehydes to Allenamides

Rémi Blieck, Sébastien Lemouzy, Arie van Der Lee, Marc Taillefer and Florian Monnier
Organic Letters
15/11/2021

Abstract

Synergistic catalysis α-Addition Allenes Copper Enamine
We herein describe an intermolecular enantioselective α-addition of aldehydes to allenamides, using a dual copper / enamine catalytic system. Highly enantioselective addition of aldehydes were obtained thanks to secondary amine catalysts. The process was found to be highly regio-, stereo-and enantio-selective under mild conditions.
url
Find in HALView

Metrics

1 Record Views

Details

Logo image