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Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4
Article de revue   Avec comité de lecture

Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4

Christo Christov, Patricia González-Bulnes, Fanny Malhaire, Tatyana Karabencheva, Cyril Goudet, Jean-Philippe Pin, Amadeu Llebaria et Jesús Giraldo
ChemMedChem, Vol.6(1), pp.131-140
03/01/2011
PMID: 21132834

Résumé

allosteric modulators computational chemistry enantioselectivity G-protein-coupled receptors mGluR4

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