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Inactivation of Focal Adhesion Kinase FAK Rapidly Abrogates Keratinocyte Entry in Mitosis via Rho‐Associated Kinase, Resulting in Squamous Differentiation
Article de revue scientifique   Open Access   Avec comité de lecture

Inactivation of Focal Adhesion Kinase FAK Rapidly Abrogates Keratinocyte Entry in Mitosis via Rho‐Associated Kinase, Resulting in Squamous Differentiation

Lizbeth Contreras, Lorena García-Gaipo, Fe García-Reija, Anna Castro, Juana García-Pedrero, Thierry Lorca et Alberto Gandarillas
FASEB Journal, Vol.40(1)
11/01/2026
PMID: 41521614

Résumé

squamous carcinoma mitosis homeostasis epithelia differentiation cell fate cell adhesion Humans Mitosis Keratinocytes Cell Differentiation rho-Associated Kinases Focal Adhesion Kinase 1 Focal Adhesion Protein-Tyrosine Kinases Tumor Suppressor Protein p53 Cell Proliferation Cells, Cultured
Cell adhesion tightly controls cell proliferation and homeostasis in stratified epithelia by mechanisms that remain unclear. Focal adhesion kinase (FAK) transduces cell adhesion signals, is frequently deregulated in epithelial cancer, and it has been associated with proliferation and resistance to treatments. The mechanisms by which FAK controls the epithelial cell cycle are still intriguing. We previously unraveled a mitosis‐differentiation checkpoint that is the limiting factor in the keratinocyte cell cycle. To investigate whether FAK plays a role in this checkpoint, we inactivated the protein in normal human oral keratinocytes by specific shRNAs or by the specific inhibitor defactinib. Inactivation of FAK very rapidly and strikingly blocked entry into mitosis and triggered a differentiation response. This response was independent of DNA damage. Tumor suppressor P53 was induced shortly after inhibition of FAK, while mitotic Cyclin B was not translocated into the nucleus. Human epidermal N‐TERT cells that were synchronized in prometaphase failed to execute mitosis. Concomitant inhibition of FAK‐downstream Rho‐associated kinase (Rock) rescued mitotic progression. The results unveil a rapid Rock‐dependent mitosis switch upon inactivation of FAK, inducing terminal differentiation, pointing at a mitotic automatic mechanism of epithelia to suppress suprabasal proliferation of precancerous cells.

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