Logo image
Se connecter
Retour
Efficient Stereoselective Synthesis of Boron L-Amino Acid Derivatives Using Wittig and Borylation Reactions
Article de revue   Avec comité de lecture

Efficient Stereoselective Synthesis of Boron L-Amino Acid Derivatives Using Wittig and Borylation Reactions

Hassib Audi, Emmanuelle Remond, Marie-Joelle Eymin, Arnaud Tessier, Raluca Malacea-Kabbara et Sylvain Juge
Phosphorus, sulfur, and silicon and the related elements, Vol.190(5-6), pp.953-954
03/06/2015
DOI: https://doi.org/10.1080/10426507.2014.979990

Résumé

Chemistry Chemistry, Inorganic & Nuclear Chemistry, Organic Physical Sciences Science & Technology
The stereoselective synthesis of a new classes of boronato- or trifluoroborato aminoacids and peptides was described using Wittig and C-H iridium borylation as key reactions. A trifluoroborato-thiophene aminoacid derivative showed an excellent stability in aqueous conditions, useful for further applications as radiotracers by F-18 labeling.

Indicateurs

1 Consultations de la notice

Détails

Logo image