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ω-Conotoxin GVIA and dihydropyridines discriminate two types of Ca 2+ channels involved in GABA release from striatal neurons in culture
Article de revue scientifique

ω-Conotoxin GVIA and dihydropyridines discriminate two types of Ca 2+ channels involved in GABA release from striatal neurons in culture

Jean-Philippe Pin et Joël Bockaert
European journal of pharmacology. Molecular pharmacology section, Vol.188(1), p.81-84
1990

Résumé

Ca 2+ channels Dihydropyridines GABA release Striatal neurons ω-conotoxin GVIA
We previously reported that the opening of the L-type Ca 2+ channel was only partly involved in the K +-evoked Ca 2+-dependent γ-aminobutyric acid (GABA) release from striatal neurons, suggesting that probably different types of voltage-sensitive Ca 2+ channels were implicated in this physiological process. Here we demonstrate that ω-contoxin GVIA, which has been reported to block L- and N-type neuronal Ca 2+ channels, also partly inhibits the Ca 2+-dependent GABA release. The maximal effects of ω-conotoxin GVIA and nifedipine, a highly specific antagonist of the L-type channels, were additive, a total inhibition of the Ca 2+-dependent GABA release being obtained in the presence of both drugs. We therefore propose that ω-conotoxin GVIA and nifedipine block two different types of Ca 2+ channels, both involved in the GABA release process.

Indicateurs

1 Consultations de la notice

Détails

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